[CAS NO. 78617-94-4] Blue FPG-A trisodium
PRODUCTS SPECIFICATIONS [78617-94-4]
DESCRIPTION [78617-94-4]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 840.10 |
| Molecular Formula | C29H17ClN7Na3O11S3 |
| SMILES | O=S(C(C(N)=C1C2=O)=CC(NC3=CC=C(NC4=NC(Cl)=NC(NC5=CC=C(S(=O)(O[Na])=O)C=C5)=N4)C(S(=O)(O[Na])=O)=C3)=C1C(C6=C2C=CC=C6)=O)(O[Na])=O |
Summary
Blue FPG-A trisodium is a selective antagonist of P2X 1 receptor and P2Y 1 receptor with IC 50 values of 35.5 μM and 2.6 μM, respectively. Blue FPG-A trisodium is a structural isomer of the components of Reactive Blue 2 (RB2) [1] .
IC50 & Target
|
p2x1 Receptor 35.5 μM (IC 50 ) |
P2Y1 Receptor 2.6 μM (IC 50 ) |
In Vitro
Blue FPG-A trisodium (RB 2 para) (1, 3.2, 10, 32 and 100 μM) inhibits the α,β-methylene ATP (α,β-MeATP) induced contraction of the rat vas deferens (RVD) and the adenosine 5′-O-(2-thiophosphate) (ADPβS) induced relaxation of the Carbachol (HY-B1208) precontracted guinea-pig taenia coli (GPTC) [1] .
MCE has not independently confirmed the accuracy of these methods. They are for reference only.
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
