[CAS NO. 1197300-24-5] TGR5 Receptor Agonist
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PRODUCTS SPECIFICATIONS [1197300-24-5]
Store
Catalog
SLK-S0193
Brand
Selleck
CAS
1197300-24-5
DESCRIPTION [1197300-24-5]
Overview
| MDL | MFCD17169972 |
|---|---|
| Molecular Weight | 361.22 |
| Molecular Formula | C18H14Cl2N2O2 |
| SMILES | O=C(C1=C(C)ON=C1C2=CC=CC=C2Cl)N(C3=CC=C(Cl)C=C3)C |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 2.7684 mL | 13.8420 mL | 27.6840 mL |
| 5 mM | 0.5537 mL | 2.7684 mL | 5.5368 mL |
| 10 mM | 0.2768 mL | 1.3842 mL | 2.7684 mL |
| 50 mM | 0.0554 mL | 0.2768 mL | 0.5537 mL |
Description
TGR5 Receptor Agonist (TGR5, CCDC, MDK00245, compd 6) is a potent agonist of . TGR5 Receptor Agonist shows improved potency with pEC50 of 6.8 and 7.5 in the U2-OS cell assay and in melanophore cells, respectively.
In vitro
TGR5 Receptor Agonist (TGR5, CCDC, MDK00245, compd 6) shows improved potency in the U2-OS cell assay (pEC50=6.8) and in melanophore cells (pEC50=7.5).
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