[CAS NO. 959122-11-3] A922500
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PRODUCTS SPECIFICATIONS [959122-11-3]
Store
Catalog
SLK-S2674
Brand
Selleck
CAS
959122-11-3
DESCRIPTION [959122-11-3]
Overview
| MDL | MFCD12828780 |
|---|---|
| Molecular Weight | 428.48 |
| Molecular Formula | C26H24N2O4 |
| SMILES | C(=O)([C@H]1[C@H](C(O)=O)CCC1)C2=CC=C(C=C2)C3=CC=C(NC(NC4=CC=CC=C4)=O)C=C3 |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Description
A922500 (DGAT-1 Inhibitor 4a) is an inhibitor for human and mouse with of 7 nM and 24 nM, respectively, good selectivity over related acyltransferases, hERG, and a panel of anti-targets.
Features
A potent, selective, and orally bioavailable DGAT-1 inhibitor.
In vitro
A 922500 inhibits the phylogenetic family members acyl coenzyme A cholesterol acyltransferase-1 and -2 with IC50 of 296 μM. A 922500 potently inhibits huDGAT-1 and mseDGAT-1.
References
Synonyms
Cyclopentanecarboxylic acid, 2-[[4′-[[(phenylamino)carbonyl]amino][1,1′-biphenyl]-4-yl]carbonyl]-, (1R,2R)-
(1R,2R)-2-[[4′-[[(Phenylamino)carbonyl]amino][1,1′-biphenyl]-4-yl]carbonyl]cyclopentanecarboxylic acid
A 922500
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