[CAS NO. 3644-61-9]  Tolperisone HCl

Ships within Stock Price Qty Total
$0.00
$0.00
Please click "REQUEST A QUOTE" button if you need other sizes or custom synthesis
request a quote
If there is no stock, or you need other sizes or custom synthesis, please:

PRODUCTS SPECIFICATIONS [3644-61-9]

Store
Catalog
SLK-S4200
Brand
Selleck
CAS
3644-61-9

DESCRIPTION [3644-61-9]

Overview

MDLMFCD00058211
Molecular Weight281.82
Molecular FormulaC16H23NO.HCl
SMILESC(C(CN1CCCCC1)C)(=O)C2=CC=C(C)C=C2.Cl

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

1 mg5 mg10 mg
1 mM3.5484 mL17.7418 mL35.4836 mL
5 mM0.7097 mL3.5484 mL7.0967 mL
10 mM0.3548 mL1.7742 mL3.5484 mL
50 mM0.0710 mL0.3548 mL0.7097 mL

Description

Tolperisone HCl is an ion channel blocker and centrally-acting muscle relaxant.

Targets

Sodium channel [1]

In vitro

Tolperisone reduces sodium and potassium permeability in the node of Ranvier of frogs, blocks calcium currents in snail neurons and inhibits current through heterologously expressed Nav1.6 channels. Tolperisone hydrochloride represents an effective and safe treatment of painful reflex muscle spasm without the typical side effects of centrally active muscle relaxants.


Synonyms

1-Propanone, 2-methyl-1-(4-methylphenyl)-3-(1-piperidinyl)-, hydrochloride (1:1)
Propiophenone, 2,4′-dimethyl-3-piperidino-, hydrochloride
1-Propanone, 2-methyl-1-(4-methylphenyl)-3-(1-piperidinyl)-, hydrochloride
Mydocalm
1-Piperidino-2-methyl-3-(4-methylphenyl)propan-3-one hydrochloride
Tolperisone hydrochloride
Muscalm
Midocalm
Tolisartine
N 553
Isocalm
Besnoline
Kineorl
Naismeritin
Minacalm
Atmosgen
Metosomin
Menopatol
Abbsa
Arantoick
2,4′-Dimethyl-3-piperidinopropiophenone hydrochloride
Tolpidol
Tolfree
Biocalm