[CAS NO. 1210344-83-4] Ertugliflozin L-pyroglutamic acid
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PRODUCTS SPECIFICATIONS [1210344-83-4]
Store
Catalog
SLK-S4431
Brand
Selleck
CAS
1210344-83-4
DESCRIPTION [1210344-83-4]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 566 |
| Molecular Formula | C27H32ClNO10 |
| SMILES | OC[C@]12CO[C@](O2)(C3=CC(CC4=CC=C(OCC)C=C4)=C(Cl)C=C3)[C@H](O)[C@@H](O)[C@@H]1O.O=C5N[C@H](C(O)=O)CC5 |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 1.7668 mL | 8.8339 mL | 17.6678 mL |
| 5 mM | 0.3534 mL | 1.7668 mL | 3.5336 mL |
| 10 mM | 0.1767 mL | 0.8834 mL | 1.7668 mL |
| 50 mM | 0.0353 mL | 0.1767 mL | 0.3534 mL |
Description
Ertugliflozin (MK-8835, PF-04971729) L-pyroglutamic acid is a potent, selective and orally active inhibitor of the with IC50 of 0.877 nM for h-SGLT2. Ertugliflozin has the potential for the treatment of type 2 diabetes mellitus.
Targets
| h-SGLT2 [1] (Cell-free assay) |
| 0.877 nM |
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