[CAS NO. 433695-36-4] BRL-50481

Name: BRL-50481
Brand: Arctom Scientific
SKU: SLK-S5837

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PRODUCTS SPECIFICATIONS [433695-36-4]

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Catalog

SLK-S5837

Brand

Selleck

CAS

433695-36-4

DESCRIPTION [433695-36-4]

Overview

MDL	MFCD03039912
Molecular Weight	244.27
Molecular Formula	C9H12N2O4S
SMILES	S(N(C)C)(=O)(=O)C1=CC(N(=O)=O)=CC=C1C

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

Concentration Volume Mass	1 mg	5 mg	10 mg
1 mM	4.0938 mL	20.4692 mL	40.9383 mL
5 mM	0.8188 mL	4.0938 mL	8.1877 mL
10 mM	0.4094 mL	2.0469 mL	4.0938 mL
50 mM	0.0819 mL	0.4094 mL	0.8188 mL

Description

BRL-50481 is a novel and selective inhibitor of with a Ki value, derived from secondary (Dixon) plots, of 180±10 nM, being at least 200-fold selective for hrPDE7A1 over all other PDEs.

Targets

PDE7 ^[1]

References

[1] Smith SJ, et al. Mol Pharmacol. 2004, 66(6):1679-89.

Synonyms

Benzenesulfonamide, N,N,2-trimethyl-5-nitro-

N,N,2-Trimethyl-5-nitrobenzenesulfonamide

BRL 50481