[CAS NO. 739366-20-2] Anagliptin

Name: Anagliptin
Brand: Arctom Scientific
SKU: SLK-S5909

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PRODUCTS SPECIFICATIONS [739366-20-2]

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Catalog

SLK-S5909

Brand

Selleck

CAS

739366-20-2

DESCRIPTION [739366-20-2]

Overview

MDL	-
Molecular Weight	383.45
Molecular Formula	C19H25N7O2
SMILES	C(NCC(NCC(=O)N1[C@H](C#N)CCC1)(C)C)(=O)C2=CN3C(N=C2)=CC(C)=N3

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

Concentration Volume Mass	1 mg	5 mg	10 mg
1 mM	2.6079 mL	13.0395 mL	26.0790 mL
5 mM	0.5216 mL	2.6079 mL	5.2158 mL
10 mM	0.2608 mL	1.3040 mL	2.6079 mL
50 mM	0.0522 mL	0.2608 mL	0.5216 mL

Description

Anagliptin is an orally active and highly selective inhibitor and exerts anti-inflammatory effects on macrophages, adipocytes, and mouse livers by suppressing NF-κB activation.

Targets

DPP-4 ^[1]

3.3 nM

References

[1] Watanabe YS, et al. J Enzyme Inhib Med Chem. 2015, 30(6):981-8.

Synonyms

Pyrazolo[1,5-a]pyrimidine-6-carboxamide, N-[2-[[2-[(2S)-2-cyano-1-pyrrolidinyl]-2-oxoethyl]amino]-2-methylpropyl]-2-methyl-

N-[2-[[2-[(2S)-2-Cyano-1-pyrrolidinyl]-2-oxoethyl]amino]-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide

Anagliptin

Suiny

N-[2-([2-[(2S)-2-Cyanopyrrolidin-1-yl]-2-oxoethyl]amino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide