[CAS NO. 1216665-49-4] APY29
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PRODUCTS SPECIFICATIONS [1216665-49-4]
Store
Catalog
SLK-S6623
Brand
Selleck
CAS
1216665-49-4
DESCRIPTION [1216665-49-4]
Overview
| MDL | MFCD28023582 |
|---|---|
| Molecular Weight | 332.36 |
| Molecular Formula | C17H16N8 |
| SMILES | C1(NC2=CC=C3N=CNC3=C2)=NC=CC(NC4=NNC(C5CC5)=C4)=N1 |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 3.0088 mL | 15.0439 mL | 30.0879 mL |
| 5 mM | 0.6018 mL | 3.0088 mL | 6.0176 mL |
| 10 mM | 0.3009 mL | 1.5044 mL | 3.0088 mL |
| 50 mM | 0.0602 mL | 0.3009 mL | 0.6018 mL |
Description
APY29 is a type I kinase inhibitor of that binds to the ATP-binding site on IRE1α and inhibits its autophosphorylation (IC50 = 280 nM) and enhances its RNase function (EC50 = 460 nM).
Targets
| IRE1α [1] (Cell-free assay) |
| 280 nM |
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