[CAS NO. 1015787-98-0] Gefapixant
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PRODUCTS SPECIFICATIONS [1015787-98-0]
Store
Catalog
SLK-S6664
Brand
Selleck
CAS
1015787-98-0
DESCRIPTION [1015787-98-0]
Overview
| MDL | MFCD24539325 |
|---|---|
| Molecular Weight | 353.40 |
| Molecular Formula | C14H19N5O4S |
| SMILES | O=S(C1=CC(OC2=CN=C(N)N=C2N)=C(C(C)C)C=C1OC)(N)=O |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 2.8297 mL | 14.1483 mL | 28.2965 mL |
| 5 mM | 0.5659 mL | 2.8297 mL | 5.6593 mL |
| 10 mM | 0.2830 mL | 1.4148 mL | 2.8297 mL |
| 50 mM | 0.0566 mL | 0.2830 mL | 0.5659 mL |
Description
Gefapixant (AF-219, MK-7264, R1646, RG-1646, RO 4926219) is an orally active small molecule antagonist of human with IC50 of about 30 nM, 100–250 nM for and , respectively. Gefapixant has shown promise for the treatment of refractory and unexplained chronic cough.
References
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