[CAS NO. 1874276-76-2] Darovasertib (LXS-196)
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PRODUCTS SPECIFICATIONS [1874276-76-2]
Store
Catalog
SLK-S6723
Brand
Selleck
CAS
1874276-76-2
DESCRIPTION [1874276-76-2]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 472.47 |
| Molecular Formula | C22H23F3N8O |
| SMILES | O=C(C1=NC(C2=NC=CC=C2C(F)(F)F)=CN=C1N)NC3=NC=CC=C3N4CCC(C)(N)CC4 |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 2.1165 mL | 10.5827 mL | 21.1654 mL |
| 5 mM | 0.4233 mL | 2.1165 mL | 4.2331 mL |
| 10 mM | 0.2117 mL | 1.0583 mL | 2.1165 mL |
| 50 mM | 0.0423 mL | 0.2117 mL | 0.4233 mL |
Description
Darovasertib (LXS-196, IDE-196) is a selective inhibitor of .
Targets
| PKC [1] |
In vitro
LXS-196 (Darovasertib) is a highly specific PKC inhibitor that resulted in a concentration dependent inhibition of immunoprecipitated LRRK1 kinase activity, with an IC50 of ∼40 nM.
References
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