[CAS NO. 1888305-96-1]  ERK5-IN-2

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PRODUCTS SPECIFICATIONS [1888305-96-1]

Store
Catalog
SLK-S6786
Brand
Selleck
CAS
1888305-96-1

DESCRIPTION [1888305-96-1]

Overview

MDLMFCD32174287
Molecular Weight388.19
Molecular FormulaC17H11BrFN3O2
SMILESO=C(C1=CC(C(C2=C(F)C=CC=C2Br)=O)=CN1)NC3=CC=CN=C3

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

1 mg5 mg10 mg
1 mM2.5761 mL12.8803 mL25.7606 mL
5 mM0.5152 mL2.5761 mL5.1521 mL
10 mM0.2576 mL1.2880 mL2.5761 mL
50 mM0.0515 mL0.2576 mL0.5152 mL

Description

ERK5-IN-2 is an orally active, sub-micromolar, selective inhibitor with IC50 of 0.82 μM and 3 μM for ERK5 and ERK5 MEF2D, respectively.

Targets

ERK5 [1]
(Cell-free assay)
ERK5 MEF2D [1]
(Cell-free assay)
0.82 μM3 μM