[CAS NO. 2166387-65-9] BI-3802
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PRODUCTS SPECIFICATIONS [2166387-65-9]
Store
Catalog
SLK-S6937
Brand
Selleck
CAS
2166387-65-9
DESCRIPTION [2166387-65-9]
Overview
| MDL | MFCD31692350 |
|---|---|
| Molecular Weight | 484.98 |
| Molecular Formula | C24H29ClN6O3 |
| SMILES | O=C(NC)COC1=CC2=C(N(C)C1=O)C=CC(NC3=NC(N4C[C@H](C)C[C@H](C)C4)=NC=C3Cl)=C2 |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 2.0619 mL | 10.3097 mL | 20.6194 mL |
| 5 mM | 0.4124 mL | 2.0619 mL | 4.1239 mL |
| 10 mM | - | - | - |
| 50 mM | - | - | - |
Description
BI-3802 is a highly potent degrader with strong de-repression of target genes anti-proliferative effects. BI-3802 inhibits the BTB domain of BCL6 with IC50 of ≤3 nM. BI-3802 exhibits antitumor activity.
Targets
| BTB domain of BCL6 [1] (Cell-free assay) |
| 3 nM |
In vitro
BI-3802 inhibits the BTB domain of BCL6 with IC50 of ≤3 nM.
References
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