[CAS NO. 1435488-37-1] ERK5-IN-1
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PRODUCTS SPECIFICATIONS [1435488-37-1]
Store
Catalog
SLK-S7334
Brand
Selleck
CAS
1435488-37-1
DESCRIPTION [1435488-37-1]
Overview
| MDL | MFCD26142929 |
|---|---|
| Molecular Weight | 638.81 |
| Molecular Formula | C36H46N8O3 |
| SMILES | O=C1C2=C(C=CC=C2)N(C3CCCC3)C4=NC(NC5=C(OCC)C=C(C(N6CCC(N7CCN(C)CC7)CC6)=O)C=C5)=NC=C4N1C |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 1.5654 mL | 7.8271 mL | 15.6541 mL |
| 5 mM | 0.3131 mL | 1.5654 mL | 3.1308 mL |
| 10 mM | 0.1565 mL | 0.7827 mL | 1.5654 mL |
| 50 mM | 0.0313 mL | 0.1565 mL | 0.3131 mL |
Description
ERK5-IN-1 (XMD17-109) is a potent, and selective inhibitor with of 162 nM.
Targets
| ERK5 [1] |
| 162 nM |
In vitro
ERK5-IN-1 potently inhibits ERK5 biochemically with an IC50 of 162 nM and in cells with a cellular EC50 for inhibiting epidermal growth factor induced ERK5 autophosphorylation of 0.09 μM.
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