[CAS NO. 900305-37-5]  PFI-4

Ships within Stock Price Qty Total
$0.00
$0.00
Please click "REQUEST A QUOTE" button if you need other sizes or custom synthesis
request a quote
If there is no stock, or you need other sizes or custom synthesis, please:

PRODUCTS SPECIFICATIONS [900305-37-5]

Store
Catalog
SLK-S7906
Brand
Selleck
CAS
900305-37-5

DESCRIPTION [900305-37-5]

Overview

MDLMFCD14744412
Molecular Weight380.44
Molecular FormulaC21H24N4O3
SMILESO=C(NC1=C(N2CCCC2)C=C(C(N3C)=C1)N(C)C3=O)C4=CC=CC=C4OC

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

1 mg5 mg10 mg
1 mM2.6285 mL13.1427 mL26.2854 mL
5 mM0.5257 mL2.6285 mL5.2571 mL
10 mM0.2629 mL1.3143 mL2.6285 mL
50 mM---

Description

PFI-4 is a potent and selective inhibitor with of 80 nM.

Targets

BRPF1 [1]
(Cell-free assay)
BRPF2 [1]
(Cell-free assay)
BRPF3 [1]
(Cell-free assay)
80 nM7.9 μM>10μM

In vitro

PFI-4 is cell permeable, and acts by displacing the BRPF1 bromodomain from Histone H3.3.