[CAS NO. 1659305-78-8] YAP-TEAD Inhibitor 1 (Peptide 17)
Please click "REQUEST A QUOTE" button if you need other sizes or custom synthesis
request a quote
If there is no stock, or you need other sizes or custom synthesis, please:
PRODUCTS SPECIFICATIONS [1659305-78-8]
Store
Catalog
SLK-S8164
Brand
Selleck
CAS
1659305-78-8
DESCRIPTION [1659305-78-8]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 2019.86 |
| Molecular Formula | C93H144ClN23O21S2 |
| SMILES | - |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 0.4951 mL | 2.4754 mL | 4.9508 mL |
| 5 mM | 0.0990 mL | 0.4951 mL | 0.9902 mL |
| 10 mM | 0.0495 mL | 0.2475 mL | 0.4951 mL |
| 50 mM | - | - | - |
Description
YAP-TEAD Inhibitor 1 (Peptide 17) is a inhibitor which has potential usage in treatment of YAP-involved cancers with of 25 nM.
Targets
| YAP/TEAD interaction [1] (Cell-free assay) |
| 25 nM |
In vitro
The engineered peptide significantly improves the potency in disrupting YAP-TEAD interaction in vitro. This 17mer peptide demonstrates a single-digit micromolar affinity to TEAD1.
References
Powered by Arctom Copyright © 2026 Arctom. All rights
reserved.