[CAS NO. 1640294-30-9] ASP4132
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PRODUCTS SPECIFICATIONS [1640294-30-9]
Store
Catalog
SLK-S8953
Brand
Selleck
CAS
1640294-30-9
DESCRIPTION [1640294-30-9]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 937.06 |
| Molecular Formula | C46H51F3N6O8S2 |
| SMILES | O=C(C1=NC2=CC=C(C3CCN(CC4=CC=C(OC)N=C4)CC3)C=C2N1)N5CCN(CC6=CC=C(C(F)(F)F)C=C6)CC5.O=S(C7=CC=C(C)C=C7)(O)=O.O=S(C8=CC=C(C)C=C8)(O)=O |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Description
ASP4132 is a potent and orally active activator of with EC50 of 0.018 μM. ASP4132 is used as a clinical candidate for the treatment of human cancer.
Targets
| AMPK [1] (Cell-free assay) |
| 0.018 μM(EC50) |
In vitro
ASP4132 is a new type of AMPK activator with potent AMPK activation activity and attractive selective growth inhibition against human cancer cells, improves aqueous solubility, metabolic stability and animal pharmacokinetics (PK). Studies on ASP4132 have advanced to clinical trials for the treatment of cancer.
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