[CAS NO. 2556836-50-9] DGY-06-116
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PRODUCTS SPECIFICATIONS [2556836-50-9]
Store
Catalog
SLK-S9643
Brand
Selleck
CAS
2556836-50-9
DESCRIPTION [2556836-50-9]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 597.11 |
| Molecular Formula | C32H33ClN8O2 |
| SMILES | - |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 1.6747 mL | 8.3737 mL | 16.7473 mL |
| 5 mM | 0.3349 mL | 1.6747 mL | 3.3495 mL |
| 10 mM | 0.1675 mL | 0.8374 mL | 1.6747 mL |
| 50 mM | 0.0335 mL | 0.1675 mL | 0.3349 mL |
Description
DGY-06-116 is an irreversible covalent and selective inhibitor of with IC50 of 2.6 nM.
Targets
| Src [1] (Cell-free assay) |
| 2.6 nM |
In vitro
DGY-06-116 inhibits Src enzymatic activity. DGY-06-116 binds covalently to Src in a manner similar to SM1-71, where the p-loop must kink to establish the covalent bond.
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