[CAS NO. 2468015-78-1] Lufotrelvir (PF-07304814)
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PRODUCTS SPECIFICATIONS [2468015-78-1]
Store
Catalog
SLK-S9858
Brand
Selleck
CAS
2468015-78-1
DESCRIPTION [2468015-78-1]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 552.51 |
| Molecular Formula | C24H33N4O9P |
| SMILES | - |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 1.8099 mL | 9.0496 mL | 18.0992 mL |
| 5 mM | 0.3620 mL | 1.8099 mL | 3.6198 mL |
| 10 mM | 0.1810 mL | 0.9050 mL | 1.8099 mL |
| 50 mM | 0.0362 mL | 0.1810 mL | 0.3620 mL |
Targets
| SARS-CoV-2 3CLpro [1] |
| 174 nM(Ki) |
In vitro
Lufotrelvir (PF-07304814) is a phosphate prodrug of PF-00835231, and there is no statistical difference in antiviral potency of Lufotrelvir in vero cells expressing high levels of the efflux transporter P-glycoprotein, showing strong antiviral activity by inhibiting coronavirus family 3CL protease activity.[1]
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